Drug

BAY-1082439

As of the edition of 20 October 2026, BAY-1082439 is a small molecule: went quiet in 2017; acts on PIK3CA and PIK3CB.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Went quiet, 2017
Kind
Small molecule
Registered trials
1, 0 stopped early
Disease areas
Cancer

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

1 company-target row on route B and 1 company-target row on route A because of this drug.

Companies on route B for this drug

In the product

1 company-target row is on route B because of BAY-1082439.

Companies on route A for this drug

In the product

1 company-target row is on route A because of BAY-1082439.

Targets

GeneProteinUniProt
PIK3CAPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformP42336
PIK3CBPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformP42338

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 11100
All trials1

Who ran its trials

CompanyRoleYears
BayerLead sponsor of trials2012 to now