Drug

Regrelor

As of the edition of 20 October 2026, Regrelor is a small molecule: stopped in 2016; acts on P2RY12.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Stopped, 2016
Kind
Small molecule
Registered trials
2, 1 stopped early
Disease areas
Heart and blood vessels

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

1 company on route A because of this drug.

Companies on route A for this drug

In the product

1 company is on route A because of Regrelor.

Target

GeneProteinUniProt
P2RY12P2Y purinoceptor 12Q9H244

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 11100
Phase 21001
All trials2

Who ran its trials

CompanyRoleYears
Merck & Co.Lead sponsor of trials2004 to now