Drug

Sapitinib

As of the edition of 20 October 2026, Sapitinib is a small molecule: in active development; acts on EGFR, ERBB2 and ERBB3.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Active, 2014
Kind
Small molecule
Registered trials
11, 2 stopped early
Disease areas
Cancer; Skin and connective tissue; Digestive system

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

1 company-target row on route B because of this drug.

Companies on route B for this drug

In the product

1 company-target row is on route B because of Sapitinib.

Targets

GeneProteinUniProt
EGFREpidermal growth factor receptorP00533
ERBB2Receptor tyrosine-protein kinase erbB-2P04626
ERBB3Receptor tyrosine-protein kinase erbB-3P21860

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 15500
Phase 26312
All trials11

Who ran its trials

CompanyRoleYears
AstraZenecaLead sponsor of trials2008 to now