Drug

Tanzisertib

As of the edition of 20 October 2026, Tanzisertib is a small molecule: stopped in 2012; acts on MAPK10 and MAPK9.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Stopped, 2012
Kind
Small molecule
Registered trials
2, 2 stopped early
Disease areas
Lungs and airways; Skin and connective tissue

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

2 company-target rows on route A because of this drug.

Companies on route A for this drug

In the product

2 company-target rows are on route A because of Tanzisertib.

Targets

GeneProteinUniProt
MAPK9Mitogen-activated protein kinase 9P45984
MAPK10Mitogen-activated protein kinase 10P53779

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 22002
All trials2

Who ran its trials

CompanyRoleYears
Bristol Myers SquibbLead sponsor of trials2011 to now