Bexagliflozin
As of the edition of 20 October 2026, Bexagliflozin is a small molecule: marketed, first approved in 2023 (US); acts on SLC5A2; US protection ends in 2032.
Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.
The drug
- Status
- Marketed; latest approval 2023
- Kind
- Small molecule
- Brand name
- Brenzavvy
- First approved
- 20 January 2023 (US)
- Approvals on record
- 1 in 1 region
- Holder of the most recent approval
- Theracosbio
- Registered trials
- 13, 1 stopped early
- Disease areas
- Hormones; Nutrition and metabolism; Heart and blood vessels; Lungs and airways; Nervous system
US protection
US protection ends in 2032.
The last listed US drug-substance patent ends in 2032. The application that gives this date is held by Theracosbio.
This is the US only, and it is not the date generics or biosimilars can enter.
The exact date and the listings behind it
In the product5 listings count towards this date. The exact date and each listing are in the product.
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Companies that need a new molecule because of this drug
1 company on route B because of this drug.
Companies on route B for this drug
In the product1 company is on route B because of Bexagliflozin.
See the 1 company on route B for this drug, with the facts behind eachRequest access. Nothing is shown until you do.
Target
| Gene | Protein | UniProt |
|---|---|---|
| SLC5A2 | Sodium/glucose cotransporter 2 | P31639 |
Registered trials
| Phase | Trials | Completed | Active | Stopped early |
|---|---|---|---|---|
| Phase 1 | 7 | 4 | 1 | 1 |
| Phase 2 | 2 | 2 | 0 | 0 |
| Phase 3 | 3 | 2 | 0 | 0 |
| Phase 4 | 1 | 0 | 1 | 0 |
| All trials | 13 |
Who has held its approvals
| Company | Role | Years |
|---|---|---|
| Theracosbio | Originator | 2023 to now |