Drug

Derazantinib

As of the edition of 20 October 2026, Derazantinib is a small molecule: stopped in 2022; acts on FGFR1, FGFR2 and FGFR3 and 1 more.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Stopped, 2022
Kind
Small molecule
Registered trials
6, 1 stopped early
Disease areas
Cancer; Digestive system; Bones, joints and muscles; Inherited and neonatal; Pregnancy and women's health; Urinary and reproductive

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

4 company-target rows on route A because of this drug.

Companies on route A for this drug

In the product

4 company-target rows are on route A because of Derazantinib.

Targets

GeneProteinUniProt
FGFR1Fibroblast growth factor receptor 1P11362
FGFR2Fibroblast growth factor receptor 2P21802
FGFR4Fibroblast growth factor receptor 4P22455
FGFR3Fibroblast growth factor receptor 3P22607

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase not stated1000
Phase 11100
Phase 24211
All trials6

Who ran its trials

CompanyRoleYears
Basilea PharmaceuticaLead sponsor of trials2019 to now