Drug

Glesatinib

As of the edition of 20 October 2026, Glesatinib is a small molecule: stopped in 2021; acts on FLT1, FLT4 and KDR and 2 more.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Stopped, 2021
Kind
Small molecule
Registered trials
6, 2 stopped early
Disease areas
Cancer; Lungs and airways

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

4 company-target rows on route A because of this drug.

Companies on route A for this drug

In the product

4 company-target rows are on route A because of Glesatinib.

Targets

GeneProteinUniProt
METHepatocyte growth factor receptorP08581
FLT1Vascular endothelial growth factor receptor 1P17948
FLT4Vascular endothelial growth factor receptor 3P35916
KDRVascular endothelial growth factor receptor 2P35968
TEKAngiopoietin-1 receptorQ02763

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 14301
Phase 22101
All trials6

Who ran its trials

CompanyRoleYears
Bristol Myers SquibbLead sponsor of trials2008 to now