Drug

Tizaterkib

As of the edition of 20 October 2026, Tizaterkib is a small molecule: stopped in 2024; acts on MAPK1 and MAPK3.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Stopped, 2024
Kind
Small molecule
Registered trials
1, 1 stopped early
Disease areas
Blood and lymph; Cancer

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

2 company-target rows on route A because of this drug.

Companies on route A for this drug

In the product

2 company-target rows are on route A because of Tizaterkib.

Targets

GeneProteinUniProt
MAPK3Mitogen-activated protein kinase 3P27361
MAPK1Mitogen-activated protein kinase 1P28482

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 11001
All trials1

Who ran its trials

CompanyRoleYears
AntengeneLead sponsor of trials2020 to now