Drug

Zeteletinib

As of the edition of 20 October 2026, Zeteletinib is a small molecule: of no established status; acts on RET.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Status not established
Kind
Small molecule
Registered trials
1, 0 stopped early
Disease areas
Cancer; Hormones; Inherited and neonatal; Lungs and airways

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Target

GeneProteinUniProt
RETProto-oncogene tyrosine-protein kinase receptor RetP07949

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 11100
All trials1

Who ran its trials

CompanyRoleYears
Boston PharmaceuticalsLead sponsor of trials2018 to now