Drug

Celiprolol

As of the edition of 20 October 2026, Celiprolol is a small molecule: marketed, first approved in 1987 (FR); acts on ADRA2A, ADRA2B and ADRA2C and 1 more.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Marketed; latest approval 1987
Kind
Small molecule
Brand name
Celectol
First approved
5 March 1987 (FR)
Approvals on record
1 in 1 region
Holder of the most recent approval
CHEPLAPHARM ARZNEIMITTEL (ALLEMAGNE)
Registered trials
3, 0 stopped early
Disease areas
Blood and lymph; Heart and blood vessels; Inherited and neonatal; Skin and connective tissue; Lungs and airways

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Targets

GeneProteinUniProt
ADRB1Beta-1 adrenergic receptorP08588
ADRA2AAlpha-2A adrenergic receptorP08913
ADRA2BAlpha-2B adrenergic receptorP18089
ADRA2CAlpha-2C adrenergic receptorP18825

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 31010
Phase 42200
All trials3