Target

LGR4

Leucine-rich repeat-containing G protein-coupled receptor 4

As of the edition of 20 October 2026, LGR4 (leucine-rich repeat-containing G protein-coupled receptor 4, UniProt Q9BXB1) has 1 drug tested at it and 1 company on the list, 0 on route A and 0 on route B.

Sources: UniProt, ClinicalTrials.gov, ChEMBL, FDA Orange Book and Purple Book, Pharos.

The protein

UniProt
Q9BXB1
How well studied
Biology documented; no tool compounds or approved drug yet
Where it sits in the cell
At a membrane
Solved structures
23
Disease areas
Cancer; Digestive system
Registered trials of its drugs
1

Drugs at this target

StatusCount
Went quiet1
Total1
DrugStatusFurthest phaseUS protection
RosmantuzumabWent quietPhase 1none listed

1 of 1 drugs, the most tested first.

Companies at this target

Where the company standsCompanies
Undetermined1
Total on the list1