Drug

Carteolol

As of the edition of 20 October 2026, Carteolol is a small molecule: marketed, first approved in 1985 (FR); acts on ADRB1, ADRB2 and ADRB3.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Marketed; latest approval 2016
Kind
Small molecule
Brand name
Cartrol
First approved
20 February 1985 (FR)
Approvals on record
7 in 4 regions
Holder of the most recent approval
Otsuka; 5 holders in all
Registered trials
1, 0 stopped early
Disease areas
Eye

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Companies that need a new molecule because of this drug

4 company-target rows on route B because of this drug.

Companies on route B for this drug

In the product

4 company-target rows are on route B because of Carteolol.

Targets

GeneProteinUniProt
ADRB2Beta-2 adrenergic receptorP07550
ADRB1Beta-1 adrenergic receptorP08588
ADRB3Beta-3 adrenergic receptorP13945

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 41100
All trials1

Who has held its approvals

CompanyRoleYears
GSKLater holder1990 to now
NovartisAcquired holder2004 to now
AbbVieAcquired holder2012 to now
OtsukaApplicant2016 to now
AbbottOriginator1988 to 2012