Target

ADRB2

Beta-2 adrenergic receptor

As of the edition of 20 October 2026, ADRB2 (beta-2 adrenergic receptor, UniProt P07550) has 64 drugs tested at it and 78 companies on the list, 8 on route A and 11 on route B.

Sources: UniProt, ClinicalTrials.gov, ChEMBL, FDA Orange Book and Purple Book, Pharos.

The protein

UniProt
P07550
How well studied
Drug target: an approved drug acts on it
Where it sits in the cell
In more than one place
Solved structures
149
Disease areas
Lungs and airways; Immune system; Heart and blood vessels; Nervous system; Eye; Cancer; Infections; Urinary and reproductive
Registered trials of its drugs
2,068

Drugs at this target

StatusCount
Marketed40
Active1
Went quiet17
Stopped3
Withdrawn from market2
Status not established1
Total64
DrugStatusFurthest phaseUS protection
EpinephrineMarketedPhase 4none listed
AlbuterolMarketedPhase 4none listed
PropranololMarketedPhase 4none listed
FormoterolMarketedPhase 4none listed
NorepinephrineMarketedPhase 4none listed
SalmeterolMarketedPhase 4none listed
CarvedilolMarketedPhase 4none listed
TimololMarketedPhase 4none listed
IndacaterolMarketedPhase 4none listed
VilanterolMarketedPhase 4none listed
OlodaterolMarketedPhase 4Ends 2027
EphedrineMarketedPhase 4none listed

12 of 64 drugs, the most tested first.

Companies at this target

Where the company standsCompanies
Route A8
Route B11
Engaged18
Undetermined41
Total on the list78
Three companies on route A or B, with the route only
CompanyRoute
Eli LillyRoute B
PfizerRoute B
OtsukaRoute B

The other 75 companies at ADRB2

In the product

78 companies in all; 75 are not named here, and no score is.

See the 78 companies at ADRB2, ranked, with the facts behind eachRequest access. Nothing is shown until you do.