Drug

Fasudil

As of the edition of 20 October 2026, Fasudil is a small molecule: stopped in 2011; acts on ROCK1 and ROCK2.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Stopped, 2011
Kind
Small molecule
Registered trials
15, 1 stopped early
Disease areas
Nervous system; Heart and blood vessels; Cancer; Nutrition and metabolism; Mental health; Urinary and reproductive

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Targets

GeneProteinUniProt
ROCK2Rho-associated protein kinase 2O75116
ROCK1Rho-associated protein kinase 1Q13464

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 212541
Phase 32110
Phase 41000
All trials15