Drug

Ezobresib

As of the edition of 20 October 2026, Ezobresib is a small molecule: in active development; acts on BRD2, BRD3 and BRD4 and 1 more.

Sources: FDA Orange Book and Purple Book, other approval registers, ClinicalTrials.gov, ChEMBL.

The drug

Status
Active, 2028
Kind
Small molecule
Registered trials
4, 0 stopped early
Disease areas
Blood and lymph; Cancer; Immune system; Heart and blood vessels; Nervous system

US protection

No US approval on record.

With no US approval on record there are no listed US patents or exclusivities.

This is the US only.

Targets

GeneProteinUniProt
BRD4Bromodomain-containing protein 4O60885
BRD2Bromodomain-containing protein 2P25440
BRD3Bromodomain-containing protein 3Q15059
BRDTBromodomain testis-specific proteinQ58F21

Registered trials

PhaseTrialsCompletedActiveStopped early
Phase 11100
Phase 23120
All trials4

Who ran its trials

CompanyRoleYears
Bristol Myers SquibbLead sponsor of trials2015 to now